nih-gov/researchfestival.nih.gov/2015/posters/molecular-ber-ep4-imaging-towards-theranostics-basal-cell-carcinoma
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<title>Molecular Ber-EP4 imaging towards theranostics for basal cell carcinoma | NIH Research Festival</title>
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<article><div class="banner banner--gray banner--compact" style="--banner-background-image: url('/sites/default/files/media/image/2021-03/2015.jpg');--banner-background-focus: 50% 50%"><div class="banner__wrapper"><div class="banner__container"><h2 class="banner__heading">NIH Research Festival</h2><div class="banner__content"><p><strong><time datetime="2015-09-16">September 16</time> <time datetime="2015-09-18">18, 2015</time></strong></p></div></div></div></div></article>
<div class="section"><div data-drupal-messages-fallback class="hidden"></div></div><main role="main"><div id="main-content" tabindex="-1"></div><div class="section"><div class="content-sidebar"><div class="content-sidebar__main"><div class="content-sidebar__main-content"><div id="block-mainpagecontent-2"><article><h1>Molecular Ber-EP4 imaging towards theranostics for basal cell carcinoma</h1><div class="schedule"><div class="schedule__label"><div class="schedule__label-text"><time datetime="2015-09-18">Friday, September 18, 2015</time>
Poster Session V
</div></div><div class="schedule__content"><div class="schedule__item"><div class="schedule__time">2:00 3:30 p.m.</div><div class="schedule__description"><p><strong>FAES Terrace</strong></p></div><div class="schedule__description"><p><strong>NINDS</strong></p></div><div class="schedule__description"><p><strong>PHARM-3</strong></p></div></div></div></div><h2>Authors</h2><ul><li>B Dasgeb</li><li>VM Diaz</li><li>TJ Rosales</li><li>DL Sackett</li><li>JR Knutson</li><li>AH Gandjbakhche</li><li>IF Brownell</li></ul><h2>Abstract</h2><p>Basal cell carcinoma (BCC) is the most common skin cancer. Differentiating benign from malignant lesions is by biopsy, incurring considerable cost and morbidity. Dermoscopy improves clinical examination; however, its utility is limited by subjective criteria, limitations of visual assessment, and lack of information beyond the surface. Deeper imaging with a wider field of view makes macro optics essential for a non-invasive image-guided diagnosis of BCC. A more economic, time efficient and less invasive diagnostic technology is needed. BerEP4 - a pan-carcinoma biomarker is expressed on 95% of BCCs. BerEP4 is not expressed on benign lesions mimicking BCC, and is expressed negligibly on normal skin epithelium. Therefore, BerEP4 is a desirable target for molecular imaging of BCC with low background noise. We used a near-infra-red (NIR) fluorophore (alexa750) labeled BerEP4 antibody (Ab) to image BerEP4 expressing tumors in Merkel and Basal cell carcinoma mice models. Sarcoma mice model (non-Ber-EP4-expressing) served as the negative control. Alexa750-anti-shigatoxin (an Ab with no target in mice) was the negative control for Ber-EP4 Ab. After IV injection of alexa750-BerEP4 we visualized Ber-EP4 expressing tumors (BCC and Merkel) in-vivo using the Bruker In-Vivo Xtreme multimodal imager. No signal was detected from sarcoma mice model or anti-shigatoxin. The ex-vivo fluorescent microscopy of excised tumors was consistent with in-vivo results. Our goal is bedside application. If successful, this technique may offer a rapid non-invasive-image-guided diagnosis, treatment and follow up for BCC, while reducing morbidities and cost. Such a platform can be applied to other skin malignancies.</p><p><strong>Scientific Focus Area</strong>: Molecular Pharmacology</p><p class="updated"><small>This page was last updated on Friday, March 26, 2021</small></p></article>
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