Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
PPO Enzyme Assay from US Patent US12123010: "Plants having increased tolerance to herbicides"
Summary
DXR Enzyme Activity Assay from US Patent US12122799: "Antibiotics for veterinary staphylococcal infections"
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
In Vitro Activity Assay from US Patent US12122780: "Pyrimidinyl group-containing tricyclic compound serving as c-Met inhibitor"
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryRelated BioAssays by Target
In Vitro Binding Affinities Assay from US Patent US12122771: "Compounds useful for treatment of substance use disorder"
Assay data:7 Active, 7 Activity ≤ 1 µM, 7 Tested
Competitive Radioligand Binding Assay from US Patent US12122750: "AT2R antagonists and uses thereof"
Assay data:6 Active, 6 Activity ≤ 1 nM, 6 Activity ≤ 1 µM, 6 Tested
Time-Resolved Fluorescence Resonance Energy Transfer (TR-FRET) Assay from US Patent US12122742: "Small molecule direct inhibitors of KEAP1-NRF2 protein-protein interaction"
Fluorescence Polarization (FP) Assay from US Patent US12122742: "Small molecule direct inhibitors of KEAP1-NRF2 protein-protein interaction"
Assay data:4 Active, 1 Activity ≤ 1 nM, 4 Activity ≤ 1 µM, 4 Tested
Competitive Binding Assay from US Patent US20240343747: "Heteroaryl compounds as inhibitors of TYK2, composition and application thereof"
Biochemical Human PDE10A Activity Assay from US Patent US20240343729: "IMIDAZOLE ORGANIC COMPOUNDS AND THEIR USE AGAINST INFLAMMATORY BOWEL DISEASE"
LATS1 Biochemical HTRF Assay from US Patent US20240343726: "PYRROLOPYRIDINE-3- AND 4-CARBOXAMIDE COMPOSITIONS AND METHODS FOR CELLULAR PROLIFERATION"
In Vitro AAK1 Enzyme Activity Assay from US Patent US20240343720: "AAK1 INHIBITOR AND USE THEREOF"
Inhibitory Activity of Compounds Against EGFR Mutant Enzyme from US Patent US20240343694: "PYRIMIDINE DERIVATIVE, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING CANCER COMPRISING SAME AS ACTIVE INGREDIENT"
Biochemical (In Vitro) Assay from US Patent US20240342186: "PYRIDINE DERIVATIVES WITH N-LINKED CYCLIC SUBSTITUENTS AS cGAS INHIBITORS"
Assay data:9 Active, 6 Activity ≤ 1 µM, 13 Tested
AlphaScreen-Based High-Throughput Screening Assay from US Patent US20240342179: "TREATMENT OF CANCERS OR NEOPLASMS BY INHIBITING KIF15"
Inhibitory Effect of Compound I on the Enzymatic Activity of PI3Kδ and PI3Kγ In Vitro from US Patent US20240342176: "PHARMACEUTICAL COMBINATION AND APPLICATION THEREOF"
TBD from US Patent US20240342139: "DEVELOPMENT AND OPTIMIZATION OF THIOCHROMENOTHIAZOLE-BASED MSUT2 INHIBITORS AS CANDIDATES FOR THE TREATMENT OF TAUOPATHY"
Assay data:1 Tested
CYP450 Enzyme Induction Study from US Patent US12116356: "N-heterocyclic five-membered ring-containing capsid protein assembly inhibitor, pharmaceutical composition thereof, and use thereof"
Assay data:2 Tested
Human 5-HT2A Binding Assay from US Patent US12116355: "Deuterated 1-piperazino-3-phenyl indanes for treatment of schizophrenia"
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
Human D2 Binding Assay from US Patent US12116355: "Deuterated 1-piperazino-3-phenyl indanes for treatment of schizophrenia"
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on